HU-243
From Infogalactic: the planetary knowledge core
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Systematic (IUPAC) name | |
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(6aR,8S,9S,10aR)-9-(hydroxymethyl)-6,6-dimethyl-3-(2-methyloctan-2-yl)-8,9-ditritio-7,8,10,10a-tetrahydro-6aH-benzo[c]chromen-1-ol
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Identifiers | |
CAS Number | 140835-18-3 ![]() |
PubChem | CID: 3081854 |
IUPHAR/BPS | 735 |
Chemical data | |
Formula | C25H40O3 |
Molecular mass | 388.30 g/mol |
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HU-243 (AM-4056) is a synthetic cannabinoid drug that is a single enantiomer of the hydrogenated derivative of the commonly used reference agonist HU-210. It is a potent agonist at both the CB1 and CB2 receptors, with a binding affinity of 0.041nM at the CB1 receptor, making it marginally more potent than HU-210, which had an affinity of 0.061nM in the same assay.[1]
See also
References
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